Synthesis and biological activity of 5-azacytosine nucleosides derived from 4-thio-2-deoxy-L-threo-pentofuranose and 4-thio-2-deoxy-D-erythro-pentofuranose.

Academic Article

Abstract

  • 1-O-Acetyl-2-deoxy-3,5-di-O-toluoyl-4-thio-D-erythro-pentofuranose and 2-deoxy-1,3,5-tri-O-acetyl-4-thio-L-threo-pentofuranose were coupled with 5-azacytosine to obtain alpha and beta anomers of nucleosides.
  • Published In

    Keywords

  • Antineoplastic Agents, Cytosine, Drug Screening Assays, Antitumor, Hepatitis B virus, Humans, Pentoses, Tumor Cells, Cultured
  • Author List

  • Cappellacci L; Tiwari KN; Montgomery JA; Secrist JA
  • Start Page

  • 613
  • End Page

  • 614
  • Volume

  • 18
  • Issue

  • 4-5